Aminalon is a drug with a nootropic effect, which is to improve metabolism, neuronal function and their blood circulation. The first drugs aimed at improving cognitive function and the functioning of the brain in general were obtained in the last century, after which their effectiveness was tested in clinical studies on focus groups.
Many drugs were found to be useless and had the same effect as the placebo. However, several drugs have proven effective, including Aminalon. The medicine is used in neurology, psychiatry and therapy due to its pronounced nootropic effect.
The drug is used in bodybuilding and sports due to its beneficial effect on the nervous system, as well as its moderate anabolic effect - the gamma-aminobutyric acid contained in the product promotes muscle growth and fat burning.
Release form
Aminalon is available in the form of tablets - 100 pieces in one package.
Mechanism of action
The main active ingredient of Aminalon is gamma-aminobutyric acid. In the body, this substance is synthesized in the subcortical parts of the brain. GABA belongs to the inhibitory mediator of the central nervous system. By interacting with specific receptors, aminobutyric acid stops the transmission of impulses through synapses. This property of the drug is used as a component of complex therapy for Parkinson's disease, Alzheimer's, epilepsy of various origins, and sleep disorders.
In addition, gamma-aminobutyric acid is involved in many metabolic reactions in the nervous tissue. Taking the drug allows you to improve the blood supply to the brain, to increase the local trophism of cells with oxygen. The medicine has a sedative effect, so it can be taken as a sedative. In some cases, the drug is prescribed for the treatment of hypertension as a component of antihypertensive therapy.
Gamma-aminobutyric acid does not have the ability to cross the blood-brain barrier. This feature explains the small therapeutic effect of the drug in comparison with anxiolytics and tranquilizers. However, a small part can pass through the protection through specialized transporter proteins.
Aminalon stimulates the release of growth hormone produced by the anterior pituitary gland. The hormone has an anabolic effect - it accelerates the growth of muscle cells and their regeneration in case of microtrauma. Growth hormone also activates protein synthesis and accelerates the burning of fat from subcutaneous tissue. Thus, taking Aminalon is indirectly involved in muscle building and weight loss.
Indications
Indications for taking Aminalon are:
- atherosclerotic lesions of the cerebral arteries - while taking the drug, the blood supply to the nervous tissue and the work of neurons improve;
- complications resulting from traumatic brain injury;
- Alzheimer's disease - Aminalon moderately improves oxygen saturation of the brain, slows down the degradation of nervous tissue, improves memory and other cognitive functions;
- Parkinson's disease as a sedative;
- insomnia;
- frequent headaches;
- mental illness, which are accompanied by a decrease in intelligence;
- polyneuropathy of alcoholic or diabetic genesis;
- the consequences of a cerebral stroke;
- arterial hypertension.
The use of Aminalon benefits athletes - the drug induces the production of growth hormone, has a sedative effect, and corrects sleep disturbances.
Contraindications
The drug is contraindicated in case of an allergic reaction or individual intolerance. It is also not recommended to use the remedy for decompensated heart and kidney diseases.
A contraindication to the use of medication is diabetes mellitus. People with this pathology should consult with an endocrinologist before using the drug. The drug promotes the production of growth hormone, which is a counter-insular hormone that increases blood glucose levels.
Method of administration of the drug and dosage
Aminalon is recommended to be consumed 30 minutes before meals. In this case, you should drink the medicine with plenty of water.
As a rule, two tablets are prescribed per day, with the first dose being small to prevent fluctuations in blood pressure. Gradually, the concentration of the agent increases to the required values over several days.
The course depends on individual characteristics, the presence of somatic diseases, their nature and characteristics of the course. On average, the duration of therapy with Aminalon is one month.
The greatest effect is recorded in the second week of taking the medication, since gamma-aminobutyric acid has a storage property, small concentrations do not cause the necessary effect.
It is correct for athletes to take the medicine immediately after training, as well as in the interval between physical activities. The maximum allowable dosage is 3 g per day.
Side effects
In case of allergy to the drug, rhinitis, conjunctivitis, skin rashes of various localization may occur. Also, with increased sensitivity to the components of the drug, abdominal pain, nausea, vomiting, and loose stools are replaced by constipation. When such symptoms appear, the remedy should be canceled. Regular intake of the medication in rare cases causes sleep disturbance, a rise in body temperature.
The most common side effect is a change in blood pressure from low to high values. Pathology is accompanied by headache, orthostatic hypotension may appear.
Overdose and consequences
Overdose is accompanied by fluctuations in blood pressure, nausea, vomiting, abdominal cramps, and frequent stools. If the maximum permissible concentration of the drug is exceeded, you should stop using it and seek medical help. In some cases, gastric lavage and further relief of symptoms are required.
Precautions and special instructions for use
Due to the fact that Aminalon can change the value of blood pressure, it is recommended to take the first drug intake under the supervision of a doctor. In the presence of hypertension and other heart diseases, it is possible to prescribe lower doses of the drug.
It is recommended to take the medication during the daytime, otherwise insomnia may appear.
You can not combine the intake of alcohol and Aminalon. Their interaction leads to the neutralization of the therapeutic effect of the drug and an increase in the severity of side effects.
Clinical studies have not proven the effect of Aminalon on reaction and concentration, therefore, while taking it, you can drive a car.
The medicine is sold over the counter without a prescription. Before using the medicine, you should consult your doctor.
Interaction with other drugs
Aminalon can not be combined with benzodiazepine drugs, barbiturates and anticonvulsants, since potentiation of the action and the development of undesirable consequences is possible.
Storage conditions and periods
According to the instructions, the shelf life is two years from the date of manufacture. The most optimal temperature regime is from +5 to +25 degrees.
It is recommended to avoid direct sunlight.
Price
A package containing 100 tablets on average costs about 200 rubles or more.
Analogs
Amilonosar is a medicine based on nicotinoyl-gamma-aminobutyric acid. The medication belongs to the group of nootropic drugs. It improves cerebral circulation, saturation of the nervous tissue with oxygen, exhibits moderate antiplatelet activity, which is used in the treatment of coronary heart disease and other pathologies.
Long-term use of the drug can reduce the severity of amnestic syndrome, has a hypnotic and sedative effect.
Phezam is a drug that contains piracetam and cinnarizine. This combination effectively increases blood flow in the brain, improves memory, speech, mental activity. Influencing the rheological properties of blood, it reduces its viscosity, which prevents or reduces the risk of thrombus formation.
The medicine is prescribed for atherosclerosis of the arteries of the brain, frequent headaches, mental disorders, organic lesions of the central nervous system. In addition, the drug has an effect on the vestibular apparatus - it reduces its excitability. This property is used to treat various labyrinthopathies.
Noofen contains aminophenylbutyric acid. The drug has a pronounced neuroregulatory effect. Noofen improves memory and mental performance, increases learning ability, endurance, productivity and ability to work.
Against the background of taking the medication, sleep is restored, the symptoms of anxiety syndrome are stopped.
Effectively used for lability of the emotional state and mental disorders. In neurology, it is used for partial relief or complete elimination of nystagmus.
Aminalon in sports and bodybuilding
Aminalon is used in sports to enhance the production of growth hormone - somatotropin. The compound has a pronounced anabolic effect. An increase in its concentration in the blood promotes the growth of muscle mass and a faster metabolism of fatty deposits in the subcutaneous tissue, and, consequently, weight loss.
A course of drug therapy is recommended a month before the competition, since the maximum effect is achieved in two weeks as gamma-aminobutyric acid accumulates in the body.
Also, the medication is used to restore sleep, reduce anxiety symptoms, feelings of fatigue and anxiety during preparation for performances. In challenging sports, Aminalon is used to improve memory and cognitive function.
Many sports nutrition companies make a product based on gamma-aminobutyric acid. The most common dietary supplements:
- GABA from Dymatize;
- GABA Trec;
- GABA Ultimate.
The price of the supplement varies from 1,000 rubles per package or more.
